2024-03-27
REL
PDBj
PDBj
PDBj
2020-08-12
2020-09-16
2020-09-16
2024-03-27
Ministry of Science and Technology (MoST, China)
2018YFA0508100
China
National Natural Science Foundation of China (NSFC)
31870724
China
human KCNQ2 in complex with ztz240
Li X
Lv D
ion channel, TRANSPORT PROTEIN
Li X
Zhang Q
Guo P
Fu J
Mei L
Lv D
Wang J
Lai D
Ye S
Yang H
Guo J
Molecular basis for ligand activation of the human KCNQ2 channel.
Cell Res.
CN
31
52
61
2021
32884139
doi:10.1038/s41422-020-00410-8
1001-0602
7cr1
FULLOVERLAP
voltage-gated potassium channel KCNQ2
voltage-gated potassium channel KCNQ2
0
1
Homo sapiens
Potassium voltage-gated channel subfamily KQT member 2
Homo sapiens
0.073627812
4
Homo sapiens
LEVO
MAGKPPKRNAFYRKLQNFLYNVLERPRGWAFIYHAYVFLLVFSCLVLSVFSTIKEYEKSSEGALYILEIVTIVVFGVEYF
VRIWAAGCCCRYRGWRGRLKFARKPFCVIDIMVLIASIAVLAAGSQGNVFATSALRSLRFLQILRMIRMDRRGGTWKLLG
SVVYAHSKELVTAWYIGFLCLILASFLVYLAEKGENDHFDTYADALWWGLITLTTIGYGDKYPQTWNGRLLAATFTLIGV
SFFALPAGILGSGFALKVQEQHRQKHFEKRRNPAAGLIQSAWRFYATNLSRTDLHSTWQYYERTVTVPMYSSQTQTYGAS
RLIPPLNQLELLRNLKSKSGLAFRKDPPPEPSPSKGSPCRGPLCGCCPGRSSQKVSLKDRVFSSPRGVAAKGKGSPQAQT
VRRSPSADQSLEDSPSKVPKSWSFGDRSRARQAFRIKGAASRQNSEEASLPGEDIVDDKSCPCEFVTEDLTPGLKVSIRA
VCVMRFLVSKRKFKESLRPYDVMDVIEQYSAGHLDMLSRIKSLQSRVDQIVGRGPAITDKDRTKGPAEAELPEDPSMMGR
LGKVEKQVLSMEKKLDFLVNIYMQRMGIPPTETEAYFGAKEPEPAPPYHSPEDSREHVDRHGCIVKIVRSSSSTGQKNFS
VEGGSSGGWSHPQFEK
O43526
N-(6-chloranylpyridin-3-yl)-4-fluoranyl-benzamide
0.000250656
4
GB9
singleParticle
particle
8.0
ETHANE
FEI TITAN KRIOS
FLOOD BEAM
BRIGHT FIELD
FIELD EMISSION GUN
300
GATAN K2 SUMMIT (4k x 4k)
1.556
1
3.4
FSC 0.143 CUT-OFF
86988
MAXIMUM LIKELIHOOD
PROJECTION MATCHING